Basic Peptide Information

DICL ID
DICL_Pep_06383
Ion Channel
Sodium channel protein type 4 subunit alpha
Peptide Function
Antagonist
Gene Name
SCN4A

Activity Data (nM)

IC50
2100 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
RDACTXXKKCKDRQAKXQRCCA
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
[CHEMBL4524508; BDBM50520483]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
129129-65-3

Experimental Conditions

pH
pH 7.4
Holding Potential (mV)
−70 mV
Temperature
18 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)

References & Disease Information

Disease
Not specified
PubChem CID
URL
Not available
PMID
Patent
Not available